5eml A 2.39 BS02 5QK A 1 Y304 Q309 L312 L319 F327 E435 E444 V503 S578 W579 F580 Y292 Q297 L300 L307 F315 E423 E432 V491 S566 W567 F568 2.1.1.320 0000387,0000785,0002039,0003714,0005515,0005634,0005654,0005694,0005737,0005794,0005829,0006325,0006338,0006353,0006355,0006479,0007088,0008168,0008327,0008469,0010468,0016274,0018216,0032259,0032922,0032991,0034709,0035097,0035243,0035246,0042054,0042118,0042802,0043021,0044020,0044027,0044877,0045596,0045892,0046982,0048026,0048511,0048714,0070372,0070888,0090161,0097421,0140938,1901796,1904992 ic50=23nM -logKd/Ki=7.64, IC50=23nM IC50=<100nM O14744 26985292 702 RVSSGRDLNCVPEIADTLGAVAKQGFDFLCMPVFHPRFKREFIQEPAKNRPGPQTRSDLLLSGRDWNTLIVGKLSPWIRPDSKVEKIRRNSEAAMLQELNFGAYLGLPAFLLPLNQEDNTNLARVLTNHIHTGHHSSMFWMRVPLVAPEDLRDDIIENAPTTHTEEYSGEEKTWMWWHNFRTLCDYSKRIAVALEIGADLPSNHVIDRWLGEPIKAAILPTSIFLTNKKGFPVLSKMHQRLIFRLLKLEVQFIITGTNHHSEKEFCSYLQYLEYLSQNRPPPNAYELFAKGYEDYLQSPLQPLMDNLESQTYEVFEKDPIKYSQYQQAIYKCLLDRVPEEEKDTNVQVLMVLGAGRGPLVNASLRAAKQADRRIKLYAVEKNPNAVVTLENWQFEEWGSQVTVVSSDMREWVAPEKADIIVSELLGSFADNELSPECLDGAQHFLKDDGVSIPGEYTSFLAPISSSKLYNEVRACREKDRDPEAQFEMPYVVRLHNFHQLSAPQPCFTFSHPNRDPMIDNNRYCTLEFPVEVNTVLHGFAGYFETVLYQDITLSIRPETHSPGMFSWFPILFPIKQPITVREGQTICVRFWRCSNSKKVWYEWAVTAPVCSAIHNPTGRSYTIGL