2b36 A 2.8 BS01 5PP A 1 G96 F97 F149 Y158 M199 G95 F96 F148 Y157 M198 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 IC50=17nM, Ki=11.8nM P9WGR1 290 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIVGGALGEEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 2b36 B 2.8 BS01 5PP B 1 G96 F97 F149 Y158 M161 G95 F96 F148 Y157 M160 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 IC50=17nM, Ki=11.8nM P9WGR1 291 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTALGEEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 2b36 C 2.8 BS01 5PP C 1 G96 F97 M103 F149 Y158 M161 G95 F96 M102 F148 Y157 M160 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 IC50=17nM, Ki=11.8nM P9WGR1 292 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 2b36 D 2.8 BS01 5PP D 1 M103 F149 Y158 M199 M102 F148 Y157 M198 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 IC50=17nM, Ki=11.8nM P9WGR1 293 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 2b36 E 2.8 BS01 5PP E 1 Y158 I215 Y157 I200 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 IC50=17nM, Ki=11.8nM P9WGR1 294 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 2b36 F 2.8 BS01 5PP F 1 G96 F97 M103 Y158 M161 G95 F96 M102 Y157 M160 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 IC50=17nM, Ki=11.8nM P9WGR1 295 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 4bng A 2.2 BS01 5PP A 1 A95 F96 Y147 Y157 S197 A198 V201 A93 F94 Y145 Y155 S195 A196 V199 Y147 Y157 M160 K164 K199 Y145 Y155 M158 K162 K197 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 Ki=0.04nM A0A0H3JLH9 23697754 1257 NLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bng B 2.2 BS01 5PP B 1 A95 Y157 M160 S197 A198 V201 A94 Y156 M159 S196 A197 V200 Y147 Y157 M160 K164 K199 Y146 Y156 M159 K163 K198 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 Ki=0.04nM A0A0H3JLH9 23697754 1257 VNLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bng C 2.2 BS01 5PP C 1 A95 Y147 Y157 S197 A198 V201 A93 Y145 Y155 S195 A196 V199 Y147 Y157 M160 K164 K199 Y145 Y155 M158 K162 K197 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 Ki=0.04nM A0A0H3JLH9 23697754 1257 NLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bng D 2.2 BS01 5PP D 1 A95 Y147 Y157 M160 S197 A198 V201 F204 A93 Y145 Y155 M158 S195 A196 V199 F202 Y147 Y157 M160 K164 K199 Y145 Y155 M158 K162 K197 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 Ki=0.04nM A0A0H3JLH9 23697754 1257 NLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bng E 2.2 BS01 5PP E 1 A95 Y147 Y157 M160 S197 A198 V201 A93 Y145 Y155 M158 S195 A196 V199 Y147 Y157 M160 K164 K199 Y145 Y155 M158 K162 K197 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 Ki=0.04nM A0A0H3JLH9 23697754 1257 NLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bng F 2.2 BS01 5PP F 1 A95 Y157 S197 A198 V201 A94 Y156 S196 A197 V200 Y147 Y157 M160 K164 K199 Y146 Y156 M159 K163 K198 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 Ki=0.04nM A0A0H3JLH9 23697754 1257 VNLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bng G 2.2 BS01 5PP G 1 Y147 Y157 S197 A198 V201 Y145 Y155 S195 A196 V199 Y147 Y157 M160 K164 K199 Y145 Y155 M158 K162 K197 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 Ki=0.04nM A0A0H3JLH9 23697754 1257 NLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bng H 2.2 BS01 5PP H 1 A95 Y147 Y157 M160 S197 A198 V201 A93 Y145 Y155 M158 S195 A196 V199 Y147 Y157 M160 K164 K199 Y145 Y155 M158 K162 K197 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 Ki=0.04nM A0A0H3JLH9 23697754 1257 NLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK