5ek9 A 2.08 BS01 5P4 A 1 W370 P371 L381 N429 V435 W23 P24 L34 N82 V88 ? -logKd/Ki=7.33, Kd=47nM Kd=47nM, IC50=2020nM, EC50=480nM P25440 29170024 501 EQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMP 5ek9 B 2.08 BS01 5P4 B 1 W370 P371 N429 V435 W23 P24 N82 V88 ? Kd=47nM, IC50=2020nM, EC50=480nM P25440 29170024 501 EQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMP