5egu A 2.21 BS01 5NQ A 1 P82 F83 Q85 V87 D88 L92 L94 N140 P36 F37 Q39 V41 D42 L46 L48 N94 ? Kd=1.4uM -logKd/Ki=5.85, Kd=1.4uM IC50=5000nM, Kd=1400nM O60885 26735842 201 NPPPPETSNPNRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5egu B 2.21 BS01 5NQ B 1 P82 F83 Q85 V87 D88 L92 L94 N140 P30 F31 Q33 V35 D36 L40 L42 N88 ? Kd=1.4uM IC50=5000nM, Kd=1400nM O60885 26735842 201 PNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5egu C 2.21 BS01 5NQ C 1 P82 F83 Q85 V87 D88 L92 L94 N140 I146 P23 F24 Q26 V28 D29 L33 L35 N81 I87 ? Kd=1.4uM IC50=5000nM, Kd=1400nM O60885 26735842 201 TNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5egu D 2.21 BS01 5NQ D 1 P82 F83 Q85 V87 D88 L92 L94 N140 I146 P40 F41 Q43 V45 D46 L50 L52 N98 I104 ? Kd=1.4uM IC50=5000nM, Kd=1400nM O60885 26735842 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT