5a5d A 1.74 BS02 5LC A 1 Q98 R118 R205 T226 H227 R249 L253 Y288 Q77 R97 R184 T205 H206 R228 L232 Y267 ? 0006826,0030288,0046872 Kd<10nM -logKd/Ki=8.00, Kd<10nM Q0P8Q4 28383577 500 AMLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTHGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAVK 5tcy A 1.9 BS01 5LC A 1 V97 Q98 R118 K121 R205 R249 Y288 V76 Q77 R97 K100 R184 R228 Y267 ? 0006826,0030288,0046872 Kd=22nM -logKd/Ki=7.66, Kd=22nM Q0P8Q4 28383577 402 AMLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTLGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAVK 5tcy B 1.9 BS01 5LC B 1 Q98 R118 K121 R205 R249 Y288 Q78 R98 K101 R185 R229 Y268 ? 0006826,0030288,0046872 Kd=22nM Q0P8Q4 28383577 402 PAMLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTLGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAV 5tcy B 1.9 BS02 5LC C 1 D39 G42 D19 G22 ? 0006826,0030288,0046872 Kd=22nM Q0P8Q4 28383577 402 PAMLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTLGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAV 5tcy C 1.9 BS01 5LC C 1 Q98 R118 K121 L191 R205 R249 Y288 Q76 R96 K99 L169 R183 R227 Y266 ? 0006826,0030288,0046872 Kd=22nM Q0P8Q4 28383577 402 MLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTLGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAVK 8baw A 1.471 BS02 5LC A 1 M89 R109 R195 P217 H218 R240 Y279 M66 R86 R172 P194 H195 R217 Y256 0006826 37428843 402 EEMTIKHQLGEAKVKKNPEKVVVFDFGVLDTLDKLGVKVTALPQMNVPKYLEKYKSSDYQNVGSLMEPDFEKLSEIKPDVIFISGRQANLYDKLKEIGPTVYIGIDTQHYWDSFTNNMKLIGQMFGKEKEVDEELANIEKQIEEVKTKAADKKALIILTTGGKVSAYGKGSRFGLIHDVLGVPAADPNLKVTNPHGQSVSFEYIAEKNPDYLFVIDRDAVVEGKPTAKQTIENALVKKTKAYQNGHIVYLDPNYWYLSGGGLTSVSEMIKQVEEGLK 8baw B 1.471 BS02 5LC B 1 M89 R109 R195 P217 H218 R240 Y279 M65 R85 R171 P193 H194 R216 Y255 0006826 37428843 402 EMTIKHQLGEAKVKKNPEKVVVFDFGVLDTLDKLGVKVTALPQMNVPKYLEKYKSSDYQNVGSLMEPDFEKLSEIKPDVIFISGRQANLYDKLKEIGPTVYIGIDTQHYWDSFTNNMKLIGQMFGKEKEVDEELANIEKQIEEVKTKAADKKALIILTTGGKVSAYGKGSRFGLIHDVLGVPAADPNLKVTNPHGQSVSFEYIAEKNPDYLFVIDRDAVVEGKPTAKQTIENALVKKTKAYQNGHIVYLDPNYWYLSGGGLTSVSEMIKQVEEGLK 8bj9 A 2.069 BS02 5LC A 1 M85 R105 R193 H215 R237 V241 Y276 M66 R86 R174 H196 R218 V222 Y257 0006826 37428843 302 EEITIKHELGETKVKKKPEKVVVFDFGVLDSLDKLGVEVTGVPKANLPSYLEKYKDSKYENVGGLMEPDFEKINEIAPDLIIISGRQANSYEKFAEIAPTVYMGIDTKNYIDSFANNMKTLGKIFGKEKEVEKELESINKQIEAVKAKAEKTSGKALIVLTTGGKVSAYGPGSRFGIIHDVLGIKPVDANIEVSTHGQSISFEYIAEKNPDYLFVVDRDAVVAGKPSAKQTIENELVKKTNAYKNNRIIYLNPNYWYLAGGGLISVAEMINEVEKGIE