5dva A 2.50004 BS01 5FL A 1 S118 Y211 R250 S95 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0008658,0008800,0017001 Kd=280uM -logKd/Ki=3.55, Kd=280uM Kd=280000nM, IC50=250000nM Q6XEC0 27165692 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5dva B 2.50004 BS01 5FL B 1 S70 S118 T209 Y211 R250 S47 S95 T186 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0008658,0008800,0017001 Kd=280uM Kd=280000nM, IC50=250000nM Q6XEC0 27165692 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5dva C 2.50004 BS01 5FL C 1 V120 T209 Y211 R250 V97 T186 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0008658,0008800,0017001 Kd=280uM Kd=280000nM, IC50=250000nM Q6XEC0 27165692 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5dva D 2.50004 BS01 5FL D 1 S118 Y211 S244 R250 S95 Y188 S221 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0008658,0008800,0017001 Kd=280uM Kd=280000nM, IC50=250000nM Q6XEC0 27165692 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP