5dts A 1.94016 BS01 5F8 A 1 S70 S118 T209 G210 Y211 R250 S46 S94 T185 G186 Y187 R226 S70 K73 S118 Y123 W157 Y211 S46 K49 S94 Y99 W133 Y187 3.5.2.6 0008658,0008800,0017001 Kd=280uM IC50=240000nM, Kd=280000nM Q6XEC0 27165692 301 WQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5dts B 1.94016 BS01 5F8 B 1 S70 T209 G210 Y211 R250 S46 T185 G186 Y187 R226 S70 K73 S118 Y123 W157 Y211 S46 K49 S94 Y99 W133 Y187 3.5.2.6 0008658,0008800,0017001 Kd=280uM IC50=240000nM, Kd=280000nM Q6XEC0 27165692 301 WQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5dts C 1.94016 BS01 5F8 C 1 S70 S118 T209 R250 S46 S94 T185 R226 S70 K73 S118 Y123 W157 Y211 S46 K49 S94 Y99 W133 Y187 3.5.2.6 0008658,0008800,0017001 Kd=280uM -logKd/Ki=3.55, Kd=280uM IC50=240000nM, Kd=280000nM Q6XEC0 27165692 301 WQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5dts D 1.94016 BS01 5F8 D 1 T209 Y211 R250 T185 Y187 R226 S70 K73 S118 Y123 W157 Y211 S46 K49 S94 Y99 W133 Y187 3.5.2.6 0008658,0008800,0017001 Kd=280uM IC50=240000nM, Kd=280000nM Q6XEC0 27165692 301 WQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 7gs2 A 1.77 BS01 5F8 A 1 P184 R188 Q192 P184 R188 Q192 2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 P0DTD1 38289714 1501 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVT