3zlx A 2.2 BS01 5EZ A 1 L74 A76 G77 A95 M143 E144 H145 M146 D152 Q153 L197 L36 A38 G39 A57 M105 E106 H107 M108 D114 Q115 L159 D190 K192 S194 N195 D208 D217 T226 D152 K154 S156 N157 D170 D179 T185 2.7.12.2 0004672,0005524,0006468 ic50=157uM -logKd/Ki=3.80, IC50=157uM IC50=157000nM Q02750 23648182 1383 ELELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMAVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFGCPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN