5dt2 A 2.3 BS01 5EV A 1 F131 S140 L143 V144 M147 D161 S164 V169 F239 V240 N241 F243 S268 S269 F114 S123 L126 V127 M130 D144 S147 V152 F222 V223 N224 F226 S251 S252 2.1.1.360 0031151,0051726 ic50=150nM -logKd/Ki=6.82, IC50=150nM IC50=150nM Q8TEK3 27563395 401 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGNTRPSTGLLRHILQQVYNHSVTDPEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKSWTGKPVSYYLHTIDRTILENYFSSLKN 5dt2 B 2.3 BS01 5EV B 1 F131 S140 L143 V144 M147 D161 S164 V169 F239 V240 N241 F243 S268 S269 F118 S127 L130 V131 M134 D148 S151 V156 F226 V227 N228 F230 S255 S256 2.1.1.360 0031151,0051726 ic50=150nM IC50=150nM Q8TEK3 27563395 401 KLELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTLNTRPSTGLLRHILQQVYNHSVTDPEKPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKVSWTGKPVSYYLHTIDRTILENYFSSLK