3fqs A 2.1 BS01 585 A 1 L377 S379 V385 A400 A451 G454 P455 L501 L15 S17 V23 A38 A84 G87 P88 L134 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K162 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.041uM -logKd/Ki=7.39, IC50=41nM EC50=10nM, IC50=41nM, Kd=19nM, Ki=30nM P43405 19220318 1 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH 3piy A 2.55 BS01 585 A 1 V416 A428 M477 G480 L528 L542 V546 V26 A38 M81 G84 L132 L146 V150 D521 A523 R525 N526 D539 F559 D125 A127 R129 N130 D143 F163 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=6.54, IC50=0.29uM Kd=190nM Q06187 21280133 1 GYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE