5csh A 1.59 BS01 54E A 1 F121 P159 V162 I164 M225 F118 P156 V159 I161 M222 D156 K158 N161 D175 P184 S194 D153 K155 N158 D172 P181 S191 2.7.11.1 0004672,0004674,0005524,0006468 Kd=270uM -logKd/Ki=3.57, Kd=270uM IC50=500000nM P68400 28451126 401 PVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5csh A 1.59 BS02 54E A 2 Y39 I69 D103 T108 A110 Y36 I66 D100 T105 A107 D156 K158 N161 D175 P184 S194 D153 K155 N158 D172 P181 S191 2.7.11.1 0004672,0004674,0005524,0006468 Kd=270uM -logKd/Ki=3.57, Kd=270uM IC50=500000nM P68400 28451126 402 PVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5csh B 1.59 BS01 54E B 1 Y136 P159 V162 I164 Y131 P154 V157 I159 D156 K158 N161 D175 P184 S194 D151 K153 N156 D170 P179 S189 2.7.11.1 0004672,0004674,0005524,0006468 Kd=270uM IC50=500000nM P68400 28451126 403 SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV 5csh B 1.59 BS02 54E B 2 W24 H183 Q186 W23 H178 Q181 D156 K158 N161 D175 P184 S194 D151 K153 N156 D170 P179 S189 2.7.11.1 0004672,0004674,0005524,0006468 Kd=270uM IC50=500000nM P68400 28451126 404 SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV