2of2 A 2.0 BS01 547 A 1 L251 A271 Y318 M319 G322 N369 L371 L21 A41 Y88 M89 G92 N139 L141 D364 R366 A368 N369 D382 A400 F402 D134 R136 A138 N139 D152 A170 F172 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.21uM -logKd/Ki=6.68, IC50=0.21uM IC50=210nM P06239 17276681 201 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT