3eej A 2.11 BS02 53R A 1 I9 V10 E32 M33 F36 S61 I62 P63 F66 I121 I7 V8 E30 M31 F34 S59 I60 P61 F64 I119 L25 W27 E32 M33 F36 L69 I118 T140 L23 W25 E30 M31 F34 L67 I116 T138 1.5.1.3 0000166,0004146,0005575,0005739,0006730,0016491,0046452,0046654,0046655,0050661 ic50=7.3nM IC50=7.3nM Q6FPH0 19152636 229 KVPVVGIVAALLPEMGIGFQGNLPWRLAKEMKYFREVTTLTNDNSKQNVVIMGRKTWESIPQKFRPLPKRINVVVSRSFDGELRKVEDGIYHSNSLRNCLTALQSSLANENKIERIYIIGGGEIYRQSMDLADHWLITKIMPLPETTIPQMDTFLQKQELEQRFYDNSDKLVDFLPSSIQLEGRLTSQEWNGELVKGLPVQEKGYQFYFTLYTKKLEHHHHHHHH 3eej B 2.11 BS02 53R B 1 I9 V10 A11 E32 M33 F36 S61 I62 P63 I121 I7 V8 A9 E30 M31 F34 S59 I60 P61 I119 L25 W27 E32 M33 F36 L69 I118 T140 L23 W25 E30 M31 F34 L67 I116 T138 1.5.1.3 0000166,0004146,0005575,0005739,0006730,0016491,0046452,0046654,0046655,0050661 ic50=7.3nM IC50=7.3nM Q6FPH0 19152636 229 KVPVVGIVAALLPEMGIGFQGNLPWRLAKEMKYFREVTTLTNDNSKQNVVIMGRKTWESIPQKFRPLPKRINVVVSRSFDGELRKVEDGIYHSNSLRNCLTALQSSLANENKIERIYIIGGGEIYRQSMDLADHWLITKIMPLPETTIPQMDTFLQKQELEQRFYDNSDKLVDFLPSSIQLEGRLTSQEWNGELVKGLPVQEKGYQFYFTLYTKKLEHHHHHHHH 3f0b X 2.1 BS02 53R X 1 L5 V6 A7 L20 D27 L28 V31 I50 L54 F92 L5 V6 A7 L20 D27 L28 V31 I50 L54 F92 0004146,0046654,0050661 ic50=0.061uM 19249312 158 TLSILVAHDLQRVIGFENQLPWHLPNDLKHVKKLSTGHTLVMGRKTFESIGKPLPNRRNVVLTSDTSFNVEGVDVIHSIEDIYQLPGHVFIFGGQTLFEEMIDKVDDMYITVIEGKFRGDTFFPPYTFEDWEVASSVEGKLDEKNTIPHTFLHLIRK 3f0u X 1.6 BS02 53R X 1 L5 V6 A7 D27 V31 M42 I50 F92 L5 V6 A7 D27 V31 M42 I50 F92 0004146,0046654,0050661 ic50=0.19uM 19249312 158 TLSILVAHDLQRVIGFENQLPWHLPNDLKHVKKLSTGHTLVMGRKTFESIGKPLPNRRNVVLTSDTSFNVEGVDVIHSIEDIYQLPGHVFIFGGQTLYEEMIDKVDDMYITVIEGKFRGDTFFPPYTFEDWEVASSVEGKLDEKNTIPHTFLHLIRK