5bml A 2.95 BS01 4TW A 1 R84 G85 F87 G88 E89 V90 A103 K105 F120 Y155 M156 A215 D216 F368 R79 G80 F82 G83 E84 V85 A98 K100 F115 Y150 M151 A210 D211 F361 D198 K200 N203 D216 T237 D193 K195 N198 D211 T232 2.7.11.1 0004672,0004674,0005524,0006468 -logKd/Ki=8.00, Ki=10nM Ki=10.0nM Q13464 26039570 501 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEETFPIPKAFVGNQLPFVGFTYYSNRRY 5bml B 2.95 BS01 4TW B 1 R84 G85 F87 G88 E89 V90 A103 K105 F120 M153 Y155 M156 D216 F368 R80 G81 F83 G84 E85 V86 A99 K101 F116 M149 Y151 M152 D212 F364 D198 K200 N203 D216 T237 D194 K196 N199 D212 T233 2.7.11.1 0004672,0004674,0005524,0006468 Ki=10.0nM Q13464 26039570 501 MSFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEEEETFPIPKAFVGNQLPFVGFTYYSN