4zlo A 2.5 BS01 4PV A 1 E315 V318 M319 N322 I327 N383 V385 H387 L405 T406 E59 V62 M63 N66 I71 N127 V129 H131 L149 T150 D389 K391 D393 N394 D407 T427 D133 K135 D137 N138 D151 T162 2.7.11.1 0004672,0005524,0006468 ic50=12uM -logKd/Ki=4.92, IC50=12uM IC50=12000nM Q13153 26191365 601 DEEILEKLRSIVSVGDPKKKYTRFEKIGQSGTVYTAMDVATGQEVAIKQMNKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATKN