4zbi A 2.5 BS01 4M6 A 1 M250 V253 F254 R263 T266 L267 F270 G271 I294 M80 V83 F84 R93 T96 L97 F100 G101 I124 ? 0042981 Ki=0.31uM -logKd/Ki=6.51, Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 4zbi B 2.5 BS01 4M6 B 1 F228 M231 M250 V253 R263 L267 F270 G271 F58 M61 M80 V83 R93 L97 F100 G101 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVED 4zbi C 2.5 BS01 4M6 C 1 F228 M250 V253 F254 R263 T266 L267 F270 G271 F58 M80 V83 F84 R93 T96 L97 F100 G101 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 4zbi D 2.5 BS01 4M6 D 1 F228 M231 M250 V253 R263 T266 L267 F270 G271 F58 M61 M80 V83 R93 T96 L97 F100 G101 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 4zbi E 2.5 BS01 4M6 E 1 F228 M250 V253 F254 R263 T266 F270 I294 F58 M80 V83 F84 R93 T96 F100 I124 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 4zbi F 2.5 BS01 4M6 F 1 F228 M231 M250 V253 F254 R263 T266 L267 F270 G271 F58 M61 M80 V83 F84 R93 T96 L97 F100 G101 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 4zbi G 2.5 BS01 4M6 G 1 F228 M250 V253 F254 R263 T266 L267 F270 G271 I294 F58 M80 V83 F84 R93 T96 L97 F100 G101 I124 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 4zbi H 2.5 BS01 4M6 H 1 F228 M231 M250 V253 F254 T266 L267 F270 G271 I294 F58 M61 M80 V83 F84 T96 L97 F100 G101 I124 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 4zbi I 2.5 BS01 4M6 I 1 F228 M231 M250 V253 R263 T266 L267 F270 G271 I294 F58 M61 M80 V83 R93 T96 L97 F100 G101 I124 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 4zbi J 2.5 BS01 4M6 J 1 M231 M250 V253 F254 R263 T266 L267 F270 I294 M61 M80 V83 F84 R93 T96 L97 F100 I124 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 4zbi K 2.5 BS01 4M6 K 1 M250 V253 F254 R263 T266 L267 F270 G271 M80 V83 F84 R93 T96 L97 F100 G101 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 4zbi L 2.5 BS01 4M6 L 1 M250 V253 F254 R263 T266 L267 F270 G271 I294 M80 V83 F84 R93 T96 L97 F100 G101 I124 ? 0042981 Ki=0.31uM Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV