3fzt A 1.95 BS01 4JZ A 1 K457 E474 M478 V487 L504 Y505 L556 G566 D567 F568 R572 K38 E55 M59 V68 L85 Y86 L137 G147 D148 F149 R153 D549 A551 R553 N554 D567 D576 L587 D130 A132 R134 N135 D148 D154 L156 2.7.10.2 0004672,0004713,0005524,0006468 ic50=637nM -logKd/Ki=6.20, IC50=637nM Q14289 19244237 999 IAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTLDNKEKFMSEAVIMKNLDHPHIVKLIGIIEEEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGLSRDELPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIA