3v0n A 1.75 BS02 4GW A 1 F121 I123 Y126 W181 R188 D211 V212 D213 F64 I66 Y69 W124 R131 D154 V155 D156 H233 G266 W300 E303 A343 H176 G209 W243 E246 A286 2.4.1.37,2.4.1.40 0005975,0016020,0016758 P16442 23836908 402 AIGEFMVSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVP 3v0n B 1.75 BS03 4GW B 1 F121 I123 Y126 W181 D211 V212 D213 F64 I66 Y69 W124 D154 V155 D156 H233 G266 W300 E303 A343 H176 G209 W243 E246 A286 2.4.1.37,2.4.1.40 0005975,0016020,0016758 P16442 23836908 403 AIGEFMVSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVP 3v0o A 1.65 BS02 4GW A 1 F121 I123 Y126 W181 V184 R188 D211 V212 D213 K346 A350 V351 F58 I60 Y63 W118 V121 R125 D148 V149 D150 K283 A287 V288 H233 G266 W300 E303 A343 H170 G203 W237 E240 A280 2.4.1.37,2.4.1.40 0005975,0016020,0016758 P16442 23836908 402 VSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVPKNHQAVRN 3v0o B 1.65 BS02 4GW B 1 F121 I123 Y126 W181 V184 R188 D211 V212 D213 K346 F58 I60 Y63 W118 V121 R125 D148 V149 D150 K283 H233 G266 W300 E303 A343 H170 G203 W237 E240 A280 2.4.1.37,2.4.1.40 0005975,0016020,0016758 P16442 23836908 402 VSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVPK 3v0p A 1.9 BS02 4GW A 1 F121 I123 Y126 W181 R188 D211 V212 D213 A350 V351 F64 I66 Y69 W124 R131 D154 V155 D156 A293 V294 H233 G266 W300 E303 A343 H176 G209 W243 E246 A286 2.4.1.37,2.4.1.40 0005975,0016020,0016758 -logKd/Ki=6.28, Ki=0.53uM P16442 23836908 402 AIGEFMVSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVPKNHQAVRN 3v0p B 1.9 BS02 4GW B 1 F121 I123 Y126 W181 V184 R188 D211 V212 D213 K346 F64 I66 Y69 W124 V127 R131 D154 V155 D156 K289 H233 G266 W300 E303 A343 H176 G209 W243 E246 A286 2.4.1.37,2.4.1.40 0005975,0016020,0016758 P16442 23836908 402 AIGEFMVSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVPK