5yp6 A 2.2 BS02 4CX A 1 Q286 L287 W317 C320 H323 L324 R364 M365 R367 A368 V376 F377 F378 F388 L391 I397 I400 Q22 L23 W53 C56 H59 L60 R100 M101 R103 A104 V112 F113 F114 F124 L127 I133 I136 ? 0003677,0004879,0005634,0006355 ic50>0.0000316M -logKd/Ki=4.60, IC50>25uM IC50=<25119nM, EC50=20nM P51449 29456799 601 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS