2hxl A 1.8 BS01 422 A 1 T14 L15 A36 L84 C87 G90 L137 T13 L14 A35 L80 C83 G86 L133 D130 K132 E134 N135 D148 T170 D126 K128 E130 N131 D144 T166 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=12nM -logKd/Ki=7.92, IC50=12nM IC50=12nM O14757 16990002 324 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRP