4igr A 2.65 BS01 3ZA A 1 Y491 P518 T520 R525 G690 A691 T692 E739 Y765 Y59 P86 T88 R93 G138 A139 T140 E187 Y213 ? 0015276,0016020 -logKd/Ki=7.20, Kd=63nM Ki=123nM P42264 23414088 901 NRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGC 4igt A 1.24 BS01 3ZA A 1 Y471 P499 T501 R506 G674 S675 T676 E726 Y753 Y61 P89 T91 R96 G141 S142 T143 E193 Y220 ? 0015276,0016020 Kd=12.8nM -logKd/Ki=7.89, Kd=12.8nM Ki=126000nM P19491 23414088 801 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECGS