4zyu A 1.95 BS02 3YA A 1 L892 F895 M896 R897 I898 L899 N913 V946 A947 V950 L85 F88 M89 R90 I91 L92 N106 V139 A140 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=1067nM -logKd/Ki=5.97, Ki=1067nM P22102 27439469 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV