4rme A 2.3 BS02 3T2 A 1 I268 A271 A272 Q275 W305 F313 R316 A327 F346 H435 L436 I24 A27 A28 Q31 W61 F69 R72 A83 F102 H191 L192 ? 0003677,0003707,0005634,0006355,0008270 Kd=9nM Kd=1210nM, EC50=22nM P19793 26331194 500 EDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP