4wnm A 2.5 BS01 3RT A 1 L377 A400 M448 M450 A451 G454 P455 K458 N499 L501 S511 D512 L18 A41 M85 M87 A88 G91 P92 K95 N136 L138 S148 D149 D494 A496 R498 N499 D512 K533 D131 A133 R135 N136 D149 K170 2.7.10.2 0004672,0004713,0005524,0006468 Ki=18nM -logKd/Ki=7.59, IC50=0.026uM P43405 26756335 701 VYEVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNH