4rg0 A 2.5 BS01 3P0 A 1 L408 G411 V416 A428 K430 Y476 M477 A478 G480 N526 L528 D539 L13 G16 V21 A33 K35 Y81 M82 A83 G85 N131 L133 D144 D521 A523 R525 N526 D539 F559 D126 A128 R130 N131 D144 F164 2.7.10.2 0004672,0004713,0005524,0006468 ic50=50nM -logKd/Ki=7.30, IC50=50nM IC50=50nM Q06187 25466710 701 EIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREARHAFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASAAVYTIMYSCWHEKADERPTFKILLSNILDVMDEE