3fzr A 2.7 BS01 3JZ A 1 L431 G432 V439 M502 E503 L504 Y505 G508 E509 L556 L13 G14 V21 M84 E85 L86 Y87 G90 E91 L138 D549 A551 R553 N554 D567 L587 D131 A133 R135 N136 D149 L157 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=7.96, IC50=11nM IC50=31nM Q14289 19244237 999 GIAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTLDNKEKFMSEAVIMKNLDHPHIVKLIGIIEEEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGLSRTRLPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIAM