4w4v A 2.01 BS01 3H8 A 1 I70 G73 Q75 V78 A91 K93 I124 L144 M146 L148 M149 D150 A151 L206 I26 G29 Q31 V34 A47 K49 I80 L100 M102 L104 M105 D106 A107 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T182 2.7.11.24 0004672,0004707,0005524,0006468 ic50=866nM -logKd/Ki=6.94, IC50=115nM IC50=866nM P53779 25623238 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDQLDEREHTIEEWKELIYKEVMN