4u7z A 2.805 BS02 3EW A 1 K97 L118 V127 M143 D208 F209 G210 V211 S212 L215 K37 L58 V67 M83 D148 F149 G150 V151 S152 L155 D190 K192 S194 N195 D208 D217 T226 D130 K132 S134 N135 D148 D157 T165 2.7.12.2 0004672,0005524,0006468 IC50=80nM, Kd=99nM Q02750 25193232 502 MELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 7jut C 3.09 BS02 3EW C 1 K97 V127 D208 F209 S212 L215 I216 K51 V81 D162 F163 S166 L169 I170 D190 K192 N195 D208 D217 T226 D144 K146 N149 D162 D171 T180 2.7.12.2 0000165,0004672,0004674,0004708,0004713,0005515,0005524,0005634,0005737,0005739,0005769,0005770,0005813,0005816,0005856,0005925,0006468,0016020,0016310,0032872,0090170,0106310,2000641 P29678 32927473 402 ELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPMAIFELLDYIVNEPPPKLPSAVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIG 7juz C 3.21 BS02 3EW C 1 K97 L118 V127 M143 D208 F209 V211 S212 L215 K55 L76 V85 M101 D166 F167 V169 S170 L173 D190 K192 N195 D208 D217 T226 D148 K150 N153 D166 D175 T184 2.7.12.2 0000165,0004672,0004674,0004708,0004713,0005515,0005524,0005634,0005737,0005739,0005769,0005770,0005813,0005816,0005856,0005925,0006468,0016020,0016310,0032872,0090170,0106310,2000641 P29678 32927473 402 LELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMPMAIFELLDYIVNEPPPKLPSAVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 7m0t B 3.19 BS01 3EW B 1 G79 K97 M143 D208 F209 G210 V211 S212 L215 I216 M219 G38 K56 M102 D167 F168 G169 V170 S171 L174 I175 M178 D190 K192 N195 D208 D217 T226 D149 K151 N154 D167 D176 T185 2.7.12.2 0000165,0000187,0004672,0004674,0004708,0004712,0004713,0005078,0005515,0005524,0005634,0005737,0005739,0005769,0005770,0005783,0005794,0005813,0005816,0005829,0005856,0005886,0005925,0006468,0006935,0007165,0007507,0008285,0010628,0014044,0016020,0016310,0021697,0030182,0030216,0030295,0030878,0032872,0035987,0038133,0042552,0043410,0043539,0044342,0045893,0048009,0048538,0048679,0048870,0050772,0060020,0060324,0060425,0060440,0060502,0060674,0060711,0070371,0070374,0071902,0090170,0090398,0097110,0106310,1903226,2000641 IC50=80nM, Kd=99nM Q02750 34470822 401 LDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDAMANAFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLNQ