3peq A 2.4 BS01 3EQ A 1 V281 F282 C285 T289 H323 L330 V341 V348 I363 I364 K367 F368 H449 M453 L469 Y473 V61 F62 C65 T69 H103 L110 V121 V128 I143 I144 K147 F148 H229 M233 L249 Y253 ? 0003677,0004879,0005634,0006355 ic50=31.6nM -logKd/Ki=7.50, IC50=31.6nM Q03181 21414782 1 ADLKAFSKHIYNAYLKNFNMTKKKARSILTAPFVIHDIETLWQAEKGLVWLPPYKEISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNKDGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGDRPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRIKKTETETSLHPLLQEIYKD 3peq B 2.4 BS01 3EQ B 1 V281 F282 C285 T289 H323 L330 L339 V348 L353 I363 I364 K367 F368 H449 M453 L469 Y473 V61 F62 C65 T69 H103 L110 L119 V128 L133 I143 I144 K147 F148 H229 M233 L249 Y253 ? 0003677,0004879,0005634,0006355 ic50=31.6nM Q03181 21414782 2 ADLKAFSKHIYNAYLKNFNMTKKKARSILTAPFVIHDIETLWQAEKGLVWLPPYKEISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNKDGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGDRPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRIKKTETETSLHPLLQEIYKDMY