4r1v A 1.2 BS01 3E8 A 1 I1084 A1108 L1140 P1158 Y1159 M1160 K1161 G1163 D1164 R1208 M1211 A1221 D1222 Y1230 I30 A54 L86 P102 Y103 M104 K105 G107 D108 R152 M155 A165 D166 Y174 D1204 A1206 R1208 N1209 D1222 A1243 D148 A150 R152 N153 D166 A187 2.7.10.1 0004672,0004713,0005524,0006468 ic50<1nM -logKd/Ki=9.00, IC50<1nM IC50=<100nM P08581 25736998 1401 LSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFI 8au3 A 2.26 BS01 3E8 A 1 I1084 A1108 P1158 Y1159 M1160 K1161 D1164 R1208 M1211 A1221 D1222 Y1230 I33 A57 P107 Y108 M109 K110 D113 R157 M160 A170 D171 Y179 2.7.10.1 0004672,0004713,0005524,0006468 P08581 37806493 1401 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHY 8au3 B 2.26 BS01 3E8 B 1 I1084 A1108 P1158 Y1159 M1160 K1161 D1164 R1208 M1211 A1221 D1222 Y1230 I29 A53 P103 Y104 M105 K106 D109 R153 M156 A166 D167 Y175 2.7.10.1 0004672,0004713,0005524,0006468 P08581 37806493 1401 SALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHY 8au5 A 2.72 BS01 3E8 A 1 I1084 A1108 P1158 Y1159 M1160 K1161 D1164 R1208 M1211 A1221 Y1230 I18 A37 P79 Y80 M81 K82 D85 R129 M132 A142 Y151 2.7.10.1 0004672,0004713,0005524,0006468 P08581 37806493 1401 QHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNREVSQFLTEGIIMKDFSHPNVLSLLGICLRSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKIVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 8aw1 A 2.14 BS01 3E8 A 1 I1084 A1108 L1157 P1158 Y1159 M1160 K1161 D1164 R1208 M1211 A1221 D1222 Y1230 I19 A43 L83 P84 Y85 M86 K87 D90 R134 M137 A147 D148 Y156 2.7.10.1 0004672,0004713,0005524,0006468 P08581 37806493 1401 VQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNEVSQFLTEGIIMKDFSHPNVLSLLGICLRSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYDKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFI 8aw1 B 2.14 BS01 3E8 B 1 I1084 V1092 A1108 L1157 P1158 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 I21 V29 A42 L84 P85 Y86 M87 D91 R135 M138 A148 D149 Y157 2.7.10.1 0004672,0004713,0005524,0006468 P08581 37806493 1401 QAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDKKIHCAVKSLNRGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFI