2cgu A 2.5 BS01 3A3 A 1 L15 V23 K38 Y86 C87 L137 D148 L10 V18 K33 Y78 C79 L129 D140 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=13.4uM -logKd/Ki=4.87, IC50=13.4uM O14757 16574416 1272 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK