4u01 A 2.8 BS02 39W A 1 F43 H57 D79 D81 V132 K136 G137 S139 F154 R155 A156 A157 F43 H57 D79 D81 V132 K136 G137 S139 F154 R155 A156 A157 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 -logKd/Ki=8.46, IC50=0.0035uM Q9WMX2 26410074 301 APITAYSQQTRGLLGCIITSLTGRDRNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRAS 4u01 B 2.8 BS02 39W B 1 F43 Y56 H57 V132 L135 K136 G137 S139 F154 R155 A156 F43 Y56 H57 V132 L135 K136 G137 S139 F154 R155 A156 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Q9WMX2 26410074 301 APITAYSQQTRGLLGCIITSLTGRDRNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRAS 4u01 C 2.8 BS02 39W C 1 Q41 Y56 H57 D81 V132 K136 G137 S139 F154 R155 A157 Q41 Y56 H57 D81 V132 K136 G137 S139 F154 R155 A157 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Q9WMX2 26410074 301 APITAYSQQTRGLLGCIITSLTGRDRNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRAS 4u01 D 2.8 BS02 39W D 1 Q41 F43 Y56 H57 D81 V132 K136 G137 S139 F154 R155 A157 Q41 F43 Y56 H57 D81 V132 K136 G137 S139 F154 R155 A157 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Q9WMX2 26410074 301 APITAYSQQTRGLLGCIITSLTGRDRNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRAS 4u01 E 2.8 BS02 39W E 1 Y56 H57 Q80 D81 V132 L135 K136 G137 S139 F154 R155 Y56 H57 Q80 D81 V132 L135 K136 G137 S139 F154 R155 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Q9WMX2 26410074 301 APITAYSQQTRGLLGCIITSLTGRDRNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRAS 4u01 F 2.8 BS02 39W F 1 Q41 F43 Y56 H57 D79 D81 V132 L135 K136 G137 S139 F154 R155 A156 A157 Q41 F43 Y56 H57 D79 D81 V132 L135 K136 G137 S139 F154 R155 A156 A157 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Q9WMX2 26410074 301 APITAYSQQTRGLLGCIITSLTGRDRNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRAS 4u01 G 2.8 BS02 39W G 1 F43 Y56 H57 D81 V132 L135 K136 G137 S139 F154 R155 A156 F43 Y56 H57 D81 V132 L135 K136 G137 S139 F154 R155 A156 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Q9WMX2 26410074 301 APITAYSQQTRGLLGCIITSLTGRDRNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRAS 4u01 H 2.8 BS02 39W H 1 F43 Y56 H57 D79 D81 V132 L135 K136 G137 S139 F154 R155 A156 A157 F43 Y56 H57 D79 D81 V132 L135 K136 G137 S139 F154 R155 A156 A157 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Q9WMX2 26410074 301 APITAYSQQTRGLLGCIITSLTGRDRNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRAS 4u01 J 2.8 BS02 39W J 1 Q41 Y56 H57 Q80 D81 V132 L135 K136 G137 S139 F154 R155 Q41 Y56 H57 Q80 D81 V132 L135 K136 G137 S139 F154 R155 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Q9WMX2 26410074 301 APITAYSQQTRGLLGCIITSLTGRDRNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRAS