3bi6 A 2.2 BS01 396 A 1 I305 A326 K328 V360 N376 E377 Y378 C379 G381 G382 F433 D463 I13 A34 K36 V68 N84 E85 Y86 C87 G89 G90 F141 D151 D426 K428 D134 K136 2.7.10.2 0004672,0005524,0006468 ic50=15nM -logKd/Ki=7.82, IC50=15nM IC50=15nM P30291 18191399 901 SRYTTEFHELEKIGSGEFGSVFKCVKRLDGCIYAIKRSKKPLAGSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVLL