2hxq A 2.0 BS01 373 A 1 Q13 L15 A36 L84 E85 Y86 C87 G90 L137 Q12 L14 A35 L80 E81 Y82 C83 G86 L133 D130 K132 E134 N135 D148 T170 D126 K128 E130 N131 D144 T166 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=144nM -logKd/Ki=6.84, IC50=144nM IC50=140nM O14757 16990002 324 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRP