3hac	A	2.0	BS01	361	A	1	E205 E206 F357 S630 Y662 Y666 V711	E167 E168 F319 S592 Y624 Y628 V673	Y547 S630 Y631 D708 H740	Y509 S592 Y593 D670 H702	3.4.14.5	0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116		ic50=0.0083uM	-logKd/Ki=8.17, IC50=6.7nM	EC50=112nM, IC50=67nM	P27487	19539471	803 	TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP
3hac	B	2.0	BS01	361	B	1	E205 E206 F357 S630 Y662 Y666 V711	E167 E168 F319 S592 Y624 Y628 V673	Y547 S630 Y631 D708 H740	Y509 S592 Y593 D670 H702	3.4.14.5	0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116		ic50=0.0083uM		EC50=112nM, IC50=67nM	P27487	19539471	804 	TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP