3rtp A 2.4 BS01 34I A 1 I70 V78 A91 M146 E147 L148 M149 D150 A151 V196 L206 I25 V30 A43 M98 E99 L100 M101 D102 A103 V148 L158 D189 K191 N194 D207 T226 D141 K143 N146 D159 T163 2.7.11.24 0004672,0004707,0005524,0006468 ic50=7nM -logKd/Ki=8.15, IC50=7nM IC50=<100nM P53779 21813278 1 NQFYSVEVGDSTFTVLKRYQNLKPIGSGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPLDEREHTIEEWKELIYKEVMN