4tkf A 2.6 BS02 33C A 1 H1031 S1033 F1035 A1038 G1043 F1044 D1045 H1048 Y1050 I1059 Y1060 Y1071 H70 S72 F74 A77 G82 F83 D84 H87 Y89 I98 Y99 Y110 2.4.2.-,2.4.2.30 0003950 -logKd/Ki=6.55, IC50=0.285uM IC50=31nM Q9H2K2 25286857 1202 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tkf B 2.6 BS02 33C B 1 H1031 S1033 F1035 A1038 I1039 G1043 F1044 D1045 H1048 Y1060 Y1071 I1075 H75 S77 F79 A82 I83 G87 F88 D89 H92 Y104 Y115 I119 2.4.2.-,2.4.2.30 0003950 IC50=31nM Q9H2K2 25286857 1202 FQGSPDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tkf C 2.6 BS02 33C C 1 H1031 F1035 A1038 G1043 F1044 D1045 H1048 I1059 Y1060 Y1071 I1075 H79 F83 A86 G91 F92 D93 H96 I107 Y108 Y119 I123 2.4.2.-,2.4.2.30 0003950 IC50=31nM Q9H2K2 25286857 1202 NLYFQGSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tkf D 2.6 BS02 33C D 1 S1033 F1035 A1038 G1043 F1044 D1045 H1048 I1059 Y1060 Y1071 S69 F71 A74 G79 F80 D81 H84 I95 Y96 Y107 2.4.2.-,2.4.2.30 0003950 IC50=31nM Q9H2K2 25286857 1202 FQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRAEYVIYRGEQAYPEYLITYQIMRP