1u3r A 2.21 BS02 338 A 1 L298 E305 L339 L343 F356 I373 H475 L476 L36 E43 L77 L81 F94 I111 H206 L207 ? 0003677,0004879,0006355 ic50=5nM -logKd/Ki=8.30, IC50=5nM IC50=5nM Q92731 15456246 201 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMQDADSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNAHVL 1u3r B 2.21 BS02 338 B 1 L298 E305 L339 F356 H475 L476 L36 E43 L77 F94 H201 L202 ? 0003677,0004879,0006355 ic50=5nM IC50=5nM Q92731 15456246 202 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNAHVLR