4px6 A 1.6 BS01 2X6 A 1 A400 M448 E449 M450 A451 G454 P455 R498 L501 D512 A35 M78 E79 M80 A81 G84 P85 R128 L131 D142 D494 A496 R498 N499 D512 K533 D124 A126 R128 N129 D142 K159 2.7.10.2 0004672,0004713,0005524,0006468 ic50=4nM -logKd/Ki=8.40, IC50=4nM IC50=307nM P43405 24726806 701 YLDRKLLTLEDKELGSGNFGTVKKGYYQMVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVTDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNE