4pid A 1.59 BS02 2UQ A 1 G52 V53 Q115 A120 C122 G52 V53 Q115 A120 C122 H54 E71 Q115 C122 H54 E71 Q115 C122 3.4.22.39 0003677,0004197,0006508,0008234,0042025,0044423 -logKd/Ki=4.62, IC50=24uM P03252 25147618 302 MGSSEQELKAIVKDLGCGPYFLGTYDKRFPGFVSPHKLACAIVNTAGRETGGVHWMAFAWNPRSKTCYLFEPFGFSDQRLKQVYQFEYESLLRRSAIASSPDRCITLEKSTQSVQGPNSAACGLFCCMFLHAFANWPQTPMDHNPTMNLITGVPNSMLNSPQVQPTLRRNQEQLYSFLERHSPYFRSHSAQIRSATSFCHLKNM 6fdq A 2.3 BS01 2UQ A 1 W247 M262 L265 A266 S270 V271 S274 W276 C345 W85 M100 L103 A104 S108 V109 S112 W114 C183 3.4.22.- 0006508,0008234 -logKd/Ki=3.95, IC50=113uM B0B9A0 30028574 501 VPAWDSDIIFKCLCYFHTLYPGLIPLETFPPATIFNFKQKIISILEDKKAVLRGEPIKGPLPICCSKENYRRHLQRTTLLPVFMWYHPTPKTLSDTMQTMKQLAIKGSVGASHWLLVIVDIQARRLVYFDSLYNYVMPPENMKKELQSFAQQLDQVYPAYDSKKFSVKIAAKEVIQRGSGSSCGAWCCQFLHWYLKDPLTDALNDLPVDSVERHENLASFVQACEAAVQDLPELSWPEA 6fdq B 2.3 BS01 2UQ B 1 W247 A266 S270 V271 S274 H275 W276 G342 S343 C345 W93 A112 S116 V117 S120 H121 W122 G188 S189 C191 3.4.22.- 0006508,0008234 B0B9A0 30028574 501 RRQTIEALVPAWDSDIIFKCLCYFHTLYPGLIPLETFPPATIFNFKQKIISILEDKKAVLRGEPIKGPLPICCSKENYRRHLQRTTLLPVFMWYHPTPKTLSDTMQTMKQLAIKGSVGASHWLLVIVDIQARRLVYFDSLYNYVMPPENMKKELQSFAQQLDQVYPAYDSKKFSVKIAAKEVIQRGSGSSCGAWCCQFLHWYLKDPLTDALNDLPVDSVERHENLASFVQACEAAVQDLPELSWPEA