3fmz A 2.9 BS01 2T1 A 1 L35 F36 L37 A57 M73 G75 M88 Y90 Q98 H104 R121 L35 F36 L37 A57 M73 G75 M88 Y90 Q98 H104 R121 ? 0001654,0002639,0005501,0005515,0005576,0005615,0006094,0007507,0007601,0016918,0019841,0030277,0030324,0032024,0032526,0034632,0034633,0042572,0042593,0048562,0048706,0048738,0048807,0060044,0060059,0060065,0060068,0060157,0060347,0070062 -logKd/Ki=8.08, Ki=8.3nM IC50=15nM P02753 19147488 184 ERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIVAEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGNDDHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLARQYRLIVHNGYC 3fmz B 2.9 BS01 2T1 B 1 L35 F36 L37 A57 M73 M88 Y90 F96 H104 R121 F135 L35 F36 L37 A57 M73 M88 Y90 F96 H104 R121 F135 ? 0001654,0002639,0005501,0005515,0005576,0005615,0006094,0007507,0007601,0016918,0019841,0030277,0030324,0032024,0032526,0034632,0034633,0042572,0042593,0048562,0048706,0048738,0048807,0060044,0060059,0060065,0060068,0060157,0060347,0070062 IC50=15nM P02753 19147488 184 ERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIVAEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGNDDHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLARQYRLIVHNGYC 6qba A 1.8 BS01 2T1 A 1 L35 F36 L37 A57 M73 M88 Y90 H104 F135 L35 F36 L37 A57 M73 M88 Y90 H104 F135 ? 0001654,0002639,0005501,0005515,0005576,0005615,0006094,0007507,0007601,0016918,0019841,0030277,0030324,0032024,0032526,0034632,0034633,0042572,0042593,0048562,0048706,0048738,0048807,0060044,0060059,0060065,0060068,0060157,0060347,0070062 IC50=15nM P02753 32554495 201 ERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIVAEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGNDDHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLARQYRLIVHNGYCDG