3g1f A 2.5 BS01 2OM A 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D15 K37 D65 K67 M121 S122 P175 Q180 G197 R198 K42 D70 K72 D75 K37 D65 K67 D70 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 VDVMDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f B 2.5 BS01 2OM A 1 D75 I76 T79 D66 I67 T70 K42 D70 K72 D75 K33 D61 K63 D66 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 DVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f B 2.5 BS02 2OM B 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D11 K33 D61 K63 M117 S118 P171 Q176 G193 R194 K42 D70 K72 D75 K33 D61 K63 D66 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 DVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f C 2.5 BS01 2OM C 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D13 K35 D63 K65 M119 S120 P173 Q178 G195 R196 K42 D70 K72 D75 K35 D63 K65 D68 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 VMDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f C 2.5 BS02 2OM D 1 D75 T79 D68 T72 K42 D70 K72 D75 K35 D63 K65 D68 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 VMDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f D 2.5 BS01 2OM C 1 D75 T79 D65 T69 K42 D70 K72 D75 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f D 2.5 BS02 2OM D 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D10 K32 D60 K62 M116 S117 P170 Q175 G192 R193 K42 D70 K72 D75 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f E 2.5 BS01 2OM E 1 D20 D70 K72 M126 S127 P180 Q185 G202 R203 D12 D62 K64 M118 S119 P172 Q177 G194 R195 K42 D70 K72 D75 K34 D62 K64 D67 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 MDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f E 2.5 BS02 2OM F 1 D75 I76 T79 D67 I68 T71 K42 D70 K72 D75 K34 D62 K64 D67 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 MDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f F 2.5 BS01 2OM E 1 D75 I76 T79 D67 I68 T71 K42 D70 K72 D75 K34 D62 K64 D67 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 MDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f F 2.5 BS02 2OM F 1 D20 D70 K72 M126 S127 P180 A184 Q185 G202 R203 D12 D62 K64 M118 S119 P172 A176 Q177 G194 R195 K42 D70 K72 D75 K34 D62 K64 D67 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 MDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f G 2.5 BS01 2OM G 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D12 K34 D62 K64 M118 S119 P172 Q177 G194 R195 K42 D70 K72 D75 K34 D62 K64 D67 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 MDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f G 2.5 BS02 2OM H 1 D75 T79 D67 T71 K42 D70 K72 D75 K34 D62 K64 D67 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 MDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f H 2.5 BS01 2OM G 1 D75 I76 T79 D66 I67 T70 K42 D70 K72 D75 K33 D61 K63 D66 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 DVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f H 2.5 BS02 2OM H 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D11 K33 D61 K63 M117 S118 P171 Q176 G193 R194 K42 D70 K72 D75 K33 D61 K63 D66 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 DVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f I 2.5 BS01 2OM I 1 D20 K72 M126 G183 G202 R203 D7 K59 M113 G170 G189 R190 K42 D70 K72 D75 K29 D57 K59 D62 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 RLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f I 2.5 BS02 2OM J 1 D75 T79 D62 T66 K42 D70 K72 D75 K29 D57 K59 D62 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 RLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f J 2.5 BS01 2OM I 1 D75 I76 D68 I69 K42 D70 K72 D75 K35 D63 K65 D68 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 VMDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f J 2.5 BS02 2OM J 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D13 K35 D63 K65 M119 S120 P173 Q178 G195 R196 K42 D70 K72 D75 K35 D63 K65 D68 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 VMDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f K 2.5 BS01 2OM K 1 D20 D70 K72 M126 S127 P180 Q185 G202 R203 D11 D61 K63 M117 S118 P171 Q176 G193 R194 K42 D70 K72 D75 K33 D61 K63 D66 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 DVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f K 2.5 BS02 2OM L 1 D75 T79 D66 T70 K42 D70 K72 D75 K33 D61 K63 D66 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 DVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f L 2.5 BS01 2OM K 1 D75 T79 D66 T70 K42 D70 K72 D75 K33 D61 K63 D66 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 DVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f L 2.5 BS02 2OM L 1 D20 K42 D70 K72 M126 G183 Q185 G202 R203 D11 K33 D61 K63 M117 G174 Q176 G193 R194 K42 D70 K72 D75 K33 D61 K63 D66 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 DVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1f M 2.5 BS01 2OM M 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D12 K34 D62 K64 M118 S119 P172 Q177 G194 R195 K42 D70 K72 D75 K34 D62 K64 D67 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=100uM O26232 19435314 229 MDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL