6eo9 H 1.84 BS03 2OJ H 1 E97A I174 A190 V213 W215 G216 E217 G219 G226 F227 Y228 E94 I172 A193 V218 W220 G221 E222 G223 G231 F232 Y233 3.4.21.5 0004252,0005509,0006508,0007596 Ki=160nM -logKd/Ki=6.80, Ki=160nM P00734 25268757 307 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF