4n1u A 1.6 BS01 2GE A 1 F27 N33 F72 F74 W117 D119 D120 F139 F25 N31 F70 F72 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=5nM -logKd/Ki=8.30, IC50=5.0nM IC50=5.0nM, EC50=126nM P36639 24695224 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDT 4n1u B 1.6 BS01 2GE B 1 F27 N33 F72 F74 M81 W117 D119 D120 F139 F26 N32 F71 F73 M80 W116 D118 D119 F138 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=5nM IC50=5.0nM, EC50=126nM P36639 24695224 201 GASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDT 5hzx A 1.9 BS01 2GE A 1 F27 N33 F72 F74 M81 W117 D119 D120 F25 N31 F70 F72 M79 W115 D117 D118 3.6.1.-,3.6.1.56 0003723,0005634,0005737,0005739,0005759,0005829,0008413,0009151,0016787,0016791,0016818,0042262,0046872,0047429 ic50=2.8nM -logKd/Ki=8.55, IC50=2.8nM Q7ZWC3 26862114 201 TSKLLTLVLVVQPGRVLLGMKKRGFGAGKWNGFGGKVQTGETIEQAARRELLEESGLTVDTLHKIGNIKFEFIGETELMDVHIFRADNYEGEPAESDEMRPQWFDIDKIPFSQMWADDILWFPLMLQKKRFLGYFKFQGHDVIVEHKLDEVEDL 5hzx B 1.9 BS01 2GE B 1 F27 N33 F72 F74 M81 W117 D119 D120 F139 F25 N31 F70 F72 M79 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0003723,0005634,0005737,0005739,0005759,0005829,0008413,0009151,0016787,0016791,0016818,0042262,0046872,0047429 ic50=2.8nM Q7ZWC3 26862114 201 TSKLLTLVLVVQPGRVLLGMKKRGFGAGKWNGFGGKVQTGETIEQAARRELLEESGLTVDTLHKIGNIKFEFIGETELMDVHIFRADNYEGEPAESDEMRPQWFDIDKIPFSQMWADDILWFPLMLQKKRFLGYFKFQGHDVIVEHKLDEVEDL 5mzg A 1.85 BS01 2GE A 1 F27 N33 F72 F74 M81 W117 D119 D120 F139 F28 N34 F73 F75 M82 W118 D120 D121 F140 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=138nM -logKd/Ki=6.86, IC50=138nM P53368 29281266 201 HMSTSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADLWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVD 5mzg B 1.85 BS01 2GE B 1 F27 N33 F72 F74 W117 D119 D120 F139 F27 N33 F72 F74 W117 D119 D120 F139 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=138nM P53368 29281266 201 MSTSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADLWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREV 6ehh A 2.4 BS01 2GE A 1 L9 F27 N33 F72 F74 M81 W117 D119 D120 F139 L8 F26 N32 F71 F73 M80 W116 D118 D119 F138 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=32nM -logKd/Ki=7.49, IC50=32nM P53368 29281266 201 STSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVDS 6ehh B 2.4 BS01 2GE B 1 F27 N33 F72 F74 W117 D119 D120 F139 F25 N31 F70 F72 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=32nM P53368 29281266 201 TSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVD 6ehh C 2.4 BS01 2GE C 1 N33 F72 F74 W117 D119 D120 F139 N31 F70 F72 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=32nM P53368 29281266 201 TSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVD 6ehh D 2.4 BS01 2GE D 1 L9 F27 N33 F72 F74 M81 W117 D119 D120 F139 L7 F25 N31 F70 F72 M79 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=32nM P53368 29281266 201 TSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVDSF 6qqn B 2.301 BS02 2GE B 1 N167 F169 E200 Y202 V238 C241 N249 L252 L255 I318 I378 N165 F167 E198 Y200 V236 C239 N247 L250 L253 I311 I363 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 Q6B856 31302152 504 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA