1nd5 A 2.9 BS01 2BF A 1 R11 H12 R15 I18 R79 Y123 S175 H257 D258 T259 R11 H12 R15 I18 R79 Y123 S175 H257 D258 T259 3.1.3.2,3.1.3.48,3.1.3.5 0003993,0004725,0005515,0005576,0005615,0005634,0005737,0005764,0005765,0005771,0005829,0005886,0006144,0006629,0006772,0007040,0008253,0009117,0012506,0016020,0016311,0016787,0016791,0030141,0030175,0031985,0033265,0035577,0042131,0042802,0042803,0045177,0046085,0051930,0052642,0060090,0060168,0070062,0106411 -logKd/Ki=8.40, IC50=4nM IC50=4nM P15309 12525165 6000 KELKFVTLVFRHGDRSPIDTFPTDPIKESSWPQGFGQLTQLGMEQHYELGEYIRKRYRKFLNESYKHEQVYIRSTDVDRTLMSAMTNLAALFPPEGVSIWNPILLWQPIPVHTVPLSEDQLLYLPFRNCPRFQELESETLKSEEFQKRLHPYKDFIATLGKLSGLHGQDLFGIWSKVYDPLYCESVHNFTLPSWATEDTMTKLRELSELSLLSLYGIHKQKEKSRLQGGVLVNEILNHMKRATQIPSYKKLIMYSAHDTTVSGLQMALDVYNGLLPPYASCHLTELYFEKGEYFVEMYYRNETQHEPYPLMLPGCSPSCPLERFAELVGPVIPQDWSTECMT 1nd5 B 2.9 BS01 2BF B 1 R1010 H1011 R1014 I1017 R1078 Y1122 S1173 H1255 D1256 R11 H12 R15 I18 R79 Y123 S174 H256 D257 3.1.3.2,3.1.3.48,3.1.3.5 0003993,0004725,0005515,0005576,0005615,0005634,0005737,0005764,0005765,0005771,0005829,0005886,0006144,0006629,0006772,0007040,0008253,0009117,0012506,0016020,0016311,0016787,0016791,0030141,0030175,0031985,0033265,0035577,0042131,0042802,0042803,0045177,0046085,0051930,0052642,0060090,0060168,0070062,0106411 IC50=4nM P15309 12525165 6001 KELKFVTLVFRHGDRSPIDTFPTDPIKESSWPQGFGQLTQLGMEQHYELGEYIRKRYRKFLNESYKHEQVYIRSTDVDRTLMSAMTNLAALFPPEGVSIWNPILLWQPIPVHTVPLSEDQLLYLPFRNCPRQELESETLKSEEFQKRLHPYKDFIATLGKLSGLHGQDLFGIWSKVYDPLYCESVHNFTLPSWATEDTMTKLRELSELSLLSLYGIHKQKEKSRLQGGVLVNEILNHMKRATQIPSYKKLIMYSAHDTTVSGLQMALDVYNGLLPPYASCHLTELYFEKGEYFVEMYYRNETQHEPYPLMLPGCSPSCPLERFAELVGPVIPQDWSTECMTT 1nd5 C 2.9 BS01 2BF C 1 R2010 H2011 R2014 I2017 R2078 Y2122 S2174 H2256 D2257 T2258 R11 H12 R15 I18 R79 Y123 S175 H257 D258 T259 3.1.3.2,3.1.3.48,3.1.3.5 0003993,0004725,0005515,0005576,0005615,0005634,0005737,0005764,0005765,0005771,0005829,0005886,0006144,0006629,0006772,0007040,0008253,0009117,0012506,0016020,0016311,0016787,0016791,0030141,0030175,0031985,0033265,0035577,0042131,0042802,0042803,0045177,0046085,0051930,0052642,0060090,0060168,0070062,0106411 IC50=4nM P15309 12525165 6002 KELKFVTLVFRHGDRSPIDTFPTDPIKESSWPQGFGQLTQLGMEQHYELGEYIRKRYRKFLNESYKHEQVYIRSTDVDRTLMSAMTNLAALFPPEGVSIWNPILLWQPIPVHTVPLSEDQLLYLPFRNCPRFQELESETLKSEEFQKRLHPYKDFIATLGKLSGLHGQDLFGIWSKVYDPLYCESVHNFTLPSWATEDTMTKLRELSELSLLSLYGIHKQKEKSRLQGGVLVNEILNHMKRATQIPSYKKLIMYSAHDTTVSGLQMALDVYNGLLPPYASCHLTELYFEKGEYFVEMYYRNETQHEPYPLMLPGCSPSCPLERFAELVGPVIPQDWSTECMT 1nd5 D 2.9 BS01 2BF D 1 R3010 H3011 R3014 I3017 R3078 Y3122 S3174 D3178 H3256 D3257 R11 H12 R15 I18 R79 Y123 S175 D179 H257 D258 R3010 H3011 R3014 R3078 H3256 D3257 R11 H12 R15 R79 H257 D258 3.1.3.2,3.1.3.48,3.1.3.5 0003993,0004725,0005515,0005576,0005615,0005634,0005737,0005764,0005765,0005771,0005829,0005886,0006144,0006629,0006772,0007040,0008253,0009117,0012506,0016020,0016311,0016787,0016791,0030141,0030175,0031985,0033265,0035577,0042131,0042802,0042803,0045177,0046085,0051930,0052642,0060090,0060168,0070062,0106411 IC50=4nM P15309 12525165 6003 KELKFVTLVFRHGDRSPIDTFPTDPIKESSWPQGFGQLTQLGMEQHYELGEYIRKRYRKFLNESYKHEQVYIRSTDVDRTLMSAMTNLAALFPPEGVSIWNPILLWQPIPVHTVPLSEDQLLYLPFRNCPRFQELESETLKSEEFQKRLHPYKDFIATLGKLSGLHGQDLFGIWSKVYDPLYCESVHNFTLPSWATEDTMTKLRELSELSLLSLYGIHKQKEKSRLQGGVLVNEILNHMKRATQIPSYKKLIMYSAHDTTVSGLQMALDVYNGLLPPYASCHLTELYFEKGEYFVEMYYRNETQHEPYPLMLPGCSPSCPLERFAELVGPVIPQDWSTECMT