4mnf A 2.802 BS01 29L A 1 V471 E501 T529 W531 C532 F583 V23 E53 T81 W83 C84 F135 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S153 2.7.11.1 0004672,0005524,0006468 IC50=0.170000nM, Ki=0.130000nM P15056 25155755 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATESILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS 4mnf B 2.802 BS01 29L B 1 I463 V471 K483 E501 I527 T529 W531 C532 F583 I15 V23 K35 E53 I79 T81 W83 C84 F135 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S153 2.7.11.1 0004672,0005524,0006468 IC50=0.170000nM, Ki=0.130000nM P15056 25155755 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATESILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS 6u2h C 2.5 BS01 29L C 1 I463 V471 K483 E501 T529 W531 C532 F583 D594 I16 V24 K36 E54 T82 W84 C85 F136 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S158 2.7.11.1 0004672,0005524,0006468 IC50=0.170000nM, Ki=0.130000nM P15056 31988522 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLATVKSRGSILWMAPEVIRMQDSNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARELPKIHRSASEPSL 6u2h D 2.5 BS01 29L D 1 V471 K483 E501 T529 W531 C532 N580 F583 D594 V24 K36 E54 T82 W84 C85 N133 F136 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S166 2.7.11.1 0004672,0005524,0006468 IC50=0.170000nM, Ki=0.130000nM P15056 31988522 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLATVKSRWSGSEQLSGSILWMAPEVIRMQDSNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARELPKIHRSASEPSL 7shv A 2.88 BS01 29L A 1 V471 K483 E501 L514 T529 W531 C532 F583 D594 V23 K35 E53 L66 T81 W83 C84 F135 D146 2.7.11.1 0004672,0005524,0006468 P15056 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSL 7shv B 2.88 BS01 29L B 1 V471 K483 E501 T529 W531 C532 F583 D594 V23 K35 E53 T81 W83 C84 F135 D146 2.7.11.1 0004672,0005524,0006468 P15056 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSL 8chf A 4.25 BS01 29L A 1 S357 V363 A373 T421 W423 C424 F475 D486 S17 V23 A33 T81 W83 C84 F135 D146 2.7.11.1 0000165,0001678,0001934,0004672,0004674,0004709,0005515,0005524,0005634,0005737,0005739,0005741,0005794,0005829,0005886,0006338,0006468,0006915,0007165,0007190,0008285,0008286,0008625,0014044,0016310,0019899,0030154,0030878,0031143,0031267,0031333,0033138,0035019,0035023,0035773,0035994,0036211,0038133,0042060,0042552,0042802,0042981,0043066,0043154,0043410,0044024,0044342,0045104,0045595,0045944,0046872,0048009,0048011,0048538,0060324,0060333,0071550,0106310,1902042,1902531,2000145 P04049 38331211 701 DWEIEASEVMLSTRIGSGSFGTVYKGKWHGDVAVKILKVVDPTPEQFQAFRNEVAVLRKTRHVNILLFMGYMTKDNLAIVTQWCEGSSLYKHLHVQETKFQMFQLIDIARQTAQGMDYLHAKNIIHRDMKSNNIFLHEGLTVKIGDFGLATVKSRVEQPTGSVLWMAPEVIRMQDNNPFSFQSDVYSYGIVLYELMTGELPYSHINNRDQIIFMVGRGYASPDLSKLYKNCPKAMKRLVADCVKKVKEERPLFPQILSSIELLQHSLPKINRSASEPSLH 8chf B 4.25 BS01 29L B 1 G356 S357 V363 T421 W423 C424 F475 D486 G16 S17 V23 T81 W83 C84 F135 D146 2.7.11.1 0000165,0001678,0001934,0004672,0004674,0004709,0005515,0005524,0005634,0005737,0005739,0005741,0005794,0005829,0005886,0006338,0006468,0006915,0007165,0007190,0008285,0008286,0008625,0014044,0016310,0019899,0030154,0030878,0031143,0031267,0031333,0033138,0035019,0035023,0035773,0035994,0036211,0038133,0042060,0042552,0042802,0042981,0043066,0043154,0043410,0044024,0044342,0045104,0045595,0045944,0046872,0048009,0048011,0048538,0060324,0060333,0071550,0106310,1902042,1902531,2000145 P04049 38331211 701 DWEIEASEVMLSTRIGSGSFGTVYKGKWHGDVAVKILKVVDPTPEQFQAFRNEVAVLRKTRHVNILLFMGYMTKDNLAIVTQWCEGSSLYKHLHVQETKFQMFQLIDIARQTAQGMDYLHAKNIIHRDMKSNNIFLHEGLTVKIGDFGLATVKSRVEQPTGSVLWMAPEVIRMQDNNPFSFQSDVYSYGIVLYELMTGELPYSHINNRDQIIFMVGRGYASPDLSKLYKNCPKAMKRLVADCVKKVKEERPLFPQILSSIELLQHSLPKINRSASEPSLH