1u3q A 2.4 BS01 272 A 1 E305 M340 L476 E43 M78 L205 ? 0003677,0004879,0006355 ic50=3.5nM -logKd/Ki=8.46, IC50=3.5nM IC50=3.5nM Q92731 15456246 501 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNA 1u3q B 2.4 BS01 272 B 1 E305 M340 H475 L476 E45 M80 H205 L206 ? 0003677,0004879,0006355 ic50=3.5nM IC50=3.5nM Q92731 15456246 501 DALSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNA 1u3q C 2.4 BS01 272 C 1 E305 M340 L343 F356 H475 E43 M78 L81 F94 H204 ? 0003677,0004879,0006355 ic50=3.5nM IC50=3.5nM Q92731 15456246 501 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNA 1u3q D 2.4 BS01 272 D 1 E305 L339 M340 F356 E43 L77 M78 F94 ? 0003677,0004879,0006355 ic50=3.5nM IC50=3.5nM Q92731 15456246 501 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNA