2z4x A 1.9 BS03 252 A 1 D80 R89 L143 H144 Q147 K174 K238 D69 R78 L132 H133 Q136 K163 K219 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 Q12051 18800762 1101 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSHSLVPFINLLGIIYQIRDDYLNLKDFQMSFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIK 2z4x B 1.9 BS03 252 B 1 D80 R89 L143 H144 Q147 K174 D214 K238 D67 R76 L130 H131 Q134 K161 D198 K216 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=0.71uM Q12051 18800762 1102 KIDELINNDPVWSSQNESLISKPYNHILLKPGNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSSHSLVPFINLLGIIYQIRDDYLNLKDFQFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKND 2z4y A 2.1 BS01 252 A 1 D80 R89 L143 K174 Q211 D214 K238 D74 R83 L137 K168 Q199 D202 K222 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=0.71uM -logKd/Ki=6.15, IC50=0.71uM Q12051 18800762 1201 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSLVPFINLLGIIYQIRDDYLNLKDFQKGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKND 2z4y A 2.1 BS02 252 A 2 G40 R44 H73 R89 R90 G37 R38 H67 R83 R84 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=0.71uM -logKd/Ki=6.15, IC50=0.71uM Q12051 18800762 1202 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSLVPFINLLGIIYQIRDDYLNLKDFQKGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKND 2z4y B 2.1 BS01 252 B 1 S76 D80 R89 L143 H144 Q147 K174 Q211 D214 K238 S63 D67 R76 L130 H131 Q134 K161 Q193 D196 K214 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=0.71uM -logKd/Ki=6.15, IC50=0.71uM Q12051 18800762 1203 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSSLVPFINLLGIIYQIRDDYLNLKDFGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKN