2q5p A 2.3 BS01 241 A 1 F226 G284 C285 R288 S289 A292 I296 I326 L330 L333 I341 S342 F20 G64 C65 R68 S69 A72 I76 I106 L110 L113 I121 S122 ? 0003677,0004879,0005634,0006355 IC50=1nM, EC50=2.0nM P37231 17937915 5001 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 2q5p B 2.3 BS01 241 B 1 F226 G284 C285 R288 S289 A292 I326 Y327 M329 L330 L333 L340 I341 S342 F363 F20 G62 C63 R66 S67 A70 I104 Y105 M107 L108 L111 L118 I119 S120 F141 ? 0003677,0004879,0005634,0006355 IC50=1nM, EC50=2.0nM P37231 17937915 7001 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKSPFVIYDMNSLMMGEFKHITVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVILHPLLQEIYKD 8zfp A 2.48 BS02 241 A 1 G284 C285 R288 S289 A292 I326 Y327 M329 L330 L333 I341 S342 G67 C68 R71 S72 A75 I109 Y110 M112 L113 L116 I124 S125 P37231 502 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYK 8zfp B 2.48 BS02 241 B 1 F226 G284 C285 R288 S289 A292 I326 Y327 M329 L330 L333 I341 S342 F20 G66 C67 R70 S71 A74 I108 Y109 M111 L112 L115 I123 S124 P37231 502 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGDKSPFVIYDMNSLMMGEDKIKFKHEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTEPLLQEIYK 8zfs A 2.56 BS02 241 A 1 C285 R288 S289 A292 I326 M329 L330 I341 S342 C69 R72 S73 A76 I110 M113 L114 I125 S126 P37231 502 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKD 8zfs B 2.56 BS02 241 B 1 F226 G284 C285 R288 S289 A292 I326 Y327 L330 L340 I341 S342 F20 G64 C65 R68 S69 A72 I106 Y107 L110 L120 I121 S122 P37231 502 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGSPFVIYDMNSLMMGEDKIKFKHEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTHPLLQEIYK