2gtk A 2.1 BS02 208 A 1 I281 F282 C285 R288 S289 H323 L330 M364 H449 L469 Y473 I62 F63 C66 R69 S70 H104 L111 M145 H230 L250 Y254 ? 0003677,0004879,0005634,0006355 ic50=0.251uM -logKd/Ki=6.60, IC50=0.251uM EC50=760nM, IC50=251nM P37231 16737814 1001 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY